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Biological and Medicinal Chemistry

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Open-chain thiamine analogues as potent inhibitors of thiamine pyrophosphate (TPP)-dependent enzymes

Alex H. Y. Chan, Terence C. S. Ho, Finian James Leeper

Version 1 posted 30 May 2023

81

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Biological and Medicinal Chemistry

Working Paper

Cannabinoid-inspired inhibitors of Autotaxin

Mathias Eymery, Kim-Anh Nguyen, Shibom Basu, Jens Hausmann, Viet-Khoa Tran-Nguyen, Hans Peter Seidel, Lola Gutierrez, Ahcène Boumendjel, Andrew McCarthy

Version 1 posted 26 June 2023

105

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Biological and Medicinal Chemistry

Working Paper

Rational design of highly potent SARS-CoV-2 nsp14 methyltransferase inhibitors

Milan Stefek, Dominika Chalupska, Karel Chalupsky, Michala Zgarbova, Alexandra Dvorakova, Petra Krafcikova, Alice Shi Ming Li, Michal Sala, Milan Dejmek, Tomas Otava, Ema Chaloupecka, Masoud Vedadi, Jan Weber, Helena Mertlikova-Kaiserova, Radim Nencka

Version 1 posted 13 March 2023

311

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Biological and Medicinal Chemistry

Working Paper

A high-throughput assay for identifying diverse antagonists of the binding interaction between the ACE2 receptor and the dynamic spike proteins of SARS-CoV-2

Rachel Sammons, Amanda Bohanon, Anvinth Kowtha, Audrey Dejong, Eun Cho, Tamer Kaoud, Kevin Dalby

Version 1 posted 09 June 2022

212

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Biological and Medicinal Chemistry

Working Paper

A Chemical Chaperone That Prevents Insulin Fibrillation

Anirban Das, Yogesh Gangarde, Ishu Saraogi

Version 1 posted 13 December 2021

326

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Biological and Medicinal Chemistry

Working Paper

A Generative Deep Learning Approach for the Discovery of SARS CoV2 Protease Inhibitors

Noor Shaker, Mohamed Abou-Zleikha, Mubarak AlAmri, Youcef Mehellou

Version 1 posted 23 April 2020

1,439

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2

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Biological and Medicinal Chemistry

Working Paper

Fluorescent Probes with Unnatural Amino Acids to Monitor Proteasome Activity in Real-Time

Breanna L. Zerfas, Rachel A. Coleman, Andres Salazar Chaparro, Nathaniel J. Macatangay, Darci Trader

Version 1 posted 30 March 2020

567

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Organic Chemistry

Working Paper

Cellular Fucosylation Inhibitors Based on Fluorinated Fucose-1-Phosphates

Johan Pijnenborg, eline visser, Marek Noga, Emiel Rossing, Raisa Veizaj, Dirk J. Lefeber, Christian Büll, Thomas Boltje

Version 1 posted 10 November 2020

400

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Biological and Medicinal Chemistry

Working Paper

Theoretical Study of the anti-NCP Molecular Mechanism of Traditional Chinese Medicine Lianhua-Qingwen Formula (LQF)

Chenghao Ye, Meina Gao, Wangqiang Lin, Kunqian Yu, Peng Li, Guanghui Chen

Version 1 posted 23 March 2020

3,113

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2

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Biological and Medicinal Chemistry

Working Paper

How ATP-Competitive Inhibitors Allosterically Modulate Tyrosine Kinases That Contain a Src-like Regulatory Architecture

Linglan Fang, Jessica Vilas-Boas, sujata chakraborty, zachary potter, Ames Register, Markus Seeliger, Dustin J. Maly

Version 2 posted 23 April 2020

686

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Refine Search

25 results in Inhibitor, Sucralose in Keywords: Inhibitor, Sucralose

Open-chain thiamine analogues as potent inhibitors of thiamine pyrophosphate (TPP)-dependent enzymes

Cannabinoid-inspired inhibitors of Autotaxin

Rational design of highly potent SARS-CoV-2 nsp14 methyltransferase inhibitors

A high-throughput assay for identifying diverse antagonists of the binding interaction between the ACE2 receptor and the dynamic spike proteins of SARS-CoV-2

A Chemical Chaperone That Prevents Insulin Fibrillation

A Generative Deep Learning Approach for the Discovery of SARS CoV2 Protease Inhibitors

Fluorescent Probes with Unnatural Amino Acids to Monitor Proteasome Activity in Real-Time

Cellular Fucosylation Inhibitors Based on Fluorinated Fucose-1-Phosphates

Theoretical Study of the anti-NCP Molecular Mechanism of Traditional Chinese Medicine Lianhua-Qingwen Formula (LQF)

How ATP-Competitive Inhibitors Allosterically Modulate Tyrosine Kinases That Contain a Src-like Regulatory Architecture

25 results in Keywords: Inhibitor, Sucralose